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Chemicals
Lypressin Acetate CAS NO.50-57-7
<p>Lypressin Acetate, also known as Lysine Vasopressin, is a synthetic nonapeptide analogue of vasopressin featuring a lysine substitution at position 8. This structural modification results in a pharmacological profile characterized by potent antidiuretic and moderate vasopressor activities. Primarily utilized in research settings, it serves as a critical tool for studying V1a, V1b, and V2 receptor signaling pathwa…
SupplierGlobal Technology Co., Ltd.www.hqtechtirz.com
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TECHNICAL SPECIFICATIONS
| Item | Specification |
|---|---|
| Product Name | Lypressin Acetate |
| CAS NO. | 50-57-7 |
| Appearance | White to off-white lyophilized powder |
| Molecular Formula | C46H65N13O12S2 |
| Molecular Weight | 1056.22 g/mol |
| Purity (RP-HPLC) | ≥ 98.0% |
| Solubility | Soluble in water and acidic aqueous solutions; insoluble in organic solvents |
| Endotoxin | ≤1 EU/mg |
| Biological Activity | Potent antidiuretic and vasopressor activity; binds to V1a, V1b, and V2 receptors |
| Storage Conditions | Store at -20°C, protected from light and moisture |
| Stock Location | Stock in USA |
| MOQ | 1g |
1.MECHANISM OF ACTION
Lypressin Acetate functions as a multi-receptor agonist for the vasopressin receptor family (V1a, V1b, V2), which are G-protein coupled receptors. Its primary action involves binding to the V2 receptor in the renal collecting ducts, activating adenylate cyclase to increase cAMP production, which subsequently promotes the insertion of aquaporin-2 channels and enhances water reabsorption. Concurrently, its interaction with V1a receptors on vascular smooth muscle stimulates phospholipase C, leading to calcium mobilization and vasoconstriction. This dual-pathway mechanism underpins its research applications in modeling antidiuretic function and vascular response.
2.PRODUCT INDICATIONS
This product is intended for scientific investigation in areas including central diabetes insipidus, hemodynamic regulation, and coagulation studies. It is particularly relevant for researchers studying hormone replacement therapy for pituitary dysfunction, where it helps elucidate water-electrolyte homeostasis. Additionally, its role in vascular smooth muscle contraction makes it suitable for cardiovascular research, such as hypertension and shock models. The product is designed for use in receptor binding assays, cell-based signaling studies, and animal model development, targeting research on renal, endocrine, and cardiovascular systems.
3.CLINICAL EFFICACY OF PRODUCT
In experimental models, Lypressin Acetate demonstrates high efficacy in reducing urine output and increasing urine osmolality, effectively managing polyuria symptoms associated with vasopressin deficiency. Studies show it restores water balance with an antidiuretic activity of approximately 200-240 units/mg and exhibits significant vasopressor effects, making it a robust reference compound for preclinical efficacy comparisons. Its ability to activate both V1 and V2 receptors allows researchers to evaluate comprehensive physiological responses, including antidiuresis, vascular contraction, and potential hemostatic effects in bleeding models.
4.Certificate
GlobalTech Co., Ltd. is committed to providing high-purity biotechnological peptide products, adhering strictly to quality standards and obtaining internationally recognized certifications.
Our production partners all employ GMP-compliant production systems and possess standardized quality control processes covering raw material procurement, synthesis, purification, testing, packaging, and storage. Each batch of product comes with complete documentation, including a Certificate of Analysis (COA), HPLC purity report, mass spectrometry (MS) chromatograms, and third-party testing reports available upon request.
We prioritize:
1.A rigorous quality management system
2.Batch traceability and stability data
3.Professional laboratory testing and validation
4.Compliance with international trade standards
Our commitment to quality, transparency, and regulatory compliance ensures the provision of reliable, stable, and research-grade peptide products to our global partners.
5.DELIVERY & SHIPPING
We specialize in global logistics for various cosmetic peptides. Your order will be handled with the utmost care, ensuring safe, reliable, and intact delivery.
Professional and Secure Packaging
Each bottle of peptide is protected with a special packaging solution to ensure stability and integrity during transportation.
We can also customize packaging according to customer needs.
Shipping Methods
Main Method: International Air Freight
We primarily use DHL, FedEx, UPS, and TNT because of their global reliability, speed, and advanced tracking systems. Air freight ensures the fastest transit time and minimizes the impact of environmental factors on the product.
Global Technology Co., Ltd. is a modern and advanced enterprise specializing in the production and export of active pharmaceutical ingredients (APIs), peptides, and plant extracts. The company invests in and collaborates closely with domestic manufacturers holding GMP, DMF, and FDA certifications, as well as laboratories at renowned universities, to meet diverse customer needs ranging from gram-level to ton-level. This enables Dejurui Pharmaceutical to provide customers with more flexible and convenient access to cost-effective, high-quality products and superior services.
We focus on the research and development and supply of high-quality chemical products, strictly adhering to international standards and quality systems. Our products are stable in performance and reliable in purity, widely used in industrial manufacturing, scientific research, and the fine chemical industry. We provide solid support at every stage with a professional and responsible attitude.
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If you have any product requirements, please send an email to:info@huanqiukeji9.com;whatsapp:85246842553
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